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Ajoute:1002, Huanmao Bilding, No.105, Mengcheng Wout, Hefei Vil, 230061, Lachin

APIs ak entèmedyè
Olanzapine CAS 132539-06-1

Olanzapine CAS 132539-06-1

CAS NON: 132539-06-1
Fòmil Molekilè: C17H20N4S
Pwa molekilè: 312.43300
EINECS NON: 603-618-4
MDL NON: MFCD00866702

Pwodwi detay

Deskripsyon pwodwi:

Non pwodwi: Olanzapine CAS NON: 132539-06-1

Sinonim:

2-Methyl-4- (4-methylpiperazin-1-yl) -10H-benzo [b] thieno [2,3-e] [1,4] diazepine;

2-Methyl-4- (4-methyl-1-piperazinyl) - 10H-thieno [2,3-b] [1,5] benzodyazepin LY-170053;

Chimik& Pwopriyete fizik:

Aparans: jòn poud cristalline

Egzamen: ≥99.00%

Dansite: 1.32 g / cm3

Pwen bouyi: 462,6 ℃ nan 760 mmHg

Pwen fizyon: 195 ℃

Flash Point: 233,6 ℃

Refractive Index: 3.3

Kondisyon Depo: Sere nan veso orijinal la nan yon kote ki fè nwa fre.

Presyon vapè: 0mmHg nan 25 ℃

Enfòmasyon sou sekirite:

Deklarasyon Sekirite S22; S24 / 25

HS Kòd: 2934999090

WGK Almay: 3

Yon serotonin (5-HT2) ak dopamine (D1 / D2) reseptè antagonist ak aktivite antikolinerik. Antisikotik. Olanzapine (LY170053) se yon gwo afinite pou 5-HT2 serotonin ak D2 dopamine reseptè antagonist.IC50 Valè: Sib: 5-HT Receptor Olanzapine se yon tienobenzodiazepin ki bloke espesyalman serontonin (5-hydroxytryptamine [5-HT]) 5-HT2A ak reseptè yo dopamine D2 (Ki valè yo se 4 ak 11 nM respektivman) osi byen ke muscarinic (M1), histamine (H1), 5-HT2C, 5-HT3 a 5-HT6, adrenèrjik (α (l)), ak D4 reseptè . Antipsikotik atipik pou tretman eskizofreni. Olanzapine montre pwopriyete antikolinerjik.

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