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CAS NO: 192185-72-1
Fomil molekile: C27H22Cl2Cl2N4O
Molekile Pwa: 489.39600
EINECS NON: NA
MDL NO: MFCD0772347
Pwodwi Deskripsyon:
Non pwodwi: tipifarnib CAS NON: 192185-72-1
Sinonim:
Zarnestra;
Tipifarnib;
Tipifarnib (Zarnestra);
Chimik & Pwopriyete fizik:
Aparans: Off-blan nan pale beij solid
Assay: ≥99.0%
Dansite: 1.33g / cm3
Bouyi pwen: 681.7 ° Cat 760mMHg
Fonn Pwen: 211-213 ° C (dec.)
Flash Pwen: 366.1 ° C
Endeks refraktif: 1.671
Vapore Presyon: 1.94E-18mmHg nan 25 ° C
Yon inibite farnesyltransferase. Sansibilizasyon imen miltip selil myeloma pwotesome pa bloke degradasyon nan bortezomib (B675700)-pwovoke agresomes. Epitou yo montre yo anpeche kwasans lan nan liy selil myelomia leukemia ak selil lesemi prensipal pa pwovoke apoptosi ak selil-sik blok le konbine avek rapamycin (R124000).
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